Conformationally restrained epothilone analogues as anti-leukemic agents

Date

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Publisher

United States Patent and Trademark Office

Abstract

Description

A method for synthesizing anti-leukemic epothilone analogues includes rigidifying a region between the macrolactone ring and the aromatic side-chain. The anti-leukemic compositions are non-naturally occurring epothilone analogue that are rigidified between the macrolactone ring and the aromatic side-chain.

Keywords

514/228.2, 514/323, 540/602, 544/373, 546/147, 546/200, 548/517

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